Article

Long-term passaging of pseudo-typed SARS-CoV-2 reveals the breadth of monoclonal and bispecific antibody cocktails

Hang Ma1,2,3, Hui-fang Zong1,2,4, Jun-jun Liu1,2, Ya-li Yue1,2, Yong Ke1,2, Yun-ji Liao1,2, Hao-neng Tang1,2, Lei Wang1,2, Shu-sheng Wang5, Yun-sheng Yuan1,2, Ming-yuan Wu1,2, Yan-lin Bian1,2, Bao-hong Zhang1,2, Hai-yang Yin1,2, Hua Jiang5, Tao Sun6,7, Lei Han4, Yue-qing Xie5, Jian-wei Zhu1,2
1 Engineering Research Center of Cell and Therapeutic Antibody, Ministry of Education, Shanghai 200240, China
2 School of Pharmacy, Shanghai Jiao Tong University, Shanghai 200240, China
3 School of Pharmaceutical Sciences, Southwest University, Chongqing 400715, China
4 Jecho Institute, Co., Ltd., Shanghai 200240, China
5 Jecho Laboratories, Inc., Frederick, MD 21704, USA
6 School of Agriculture and Biology, Shanghai Jiao Tong University, Shanghai 200240, China
7 Shanghai Municipal Veterinary Key Laboratory, Shanghai 200240, China
Correspondence to: Lei Han: lei.han@jechobio.com, Yue-qing Xie: yueqing.xie@jecholabs.com, Jian-wei Zhu: jianweiz@sjtu.edu.cn,
DOI: 10.1038/s41401-022-01043-w
Received: 15 October 2022
Accepted: 13 December 2022
Advance online: 27 January 2023

Abstract

The continuous emergence of severe acute respiratory syndrome coronavirus 2 (SARS-CoV-2) variants poses challenges to the effectiveness of neutralizing antibodies. Rational design of antibody cocktails is a realizable approach addressing viral immune evasion. However, evaluating the breadth of antibody cocktails is essential for understanding the development potential. Here, based on a replication competent vesicular stomatitis virus model that incorporates the spike of SARS-CoV-2 (VSV-SARS-CoV-2), we evaluated the breadth of a number of antibody cocktails consisting of monoclonal antibodies and bispecific antibodies by long- term passaging the virus in the presence of the cocktails. Results from over two-month passaging of the virus showed that 9E12 + 10D4 + 2G1 and 7B9-9D11 + 2G1 from these cocktails were highly resistant to random mutation, and there was no breakthrough after 30 rounds of passaging. As a control, antibody REGN10933 was broken through in the third passage. Next generation sequencing was performed and several critical mutations related to viral evasion were identified. These mutations caused a decrease in neutralization efficiency, but the reduced replication rate and ACE2 susceptibility of the mutant virus suggested that they might not have the potential to become epidemic strains. The 9E12 + 10D4 + 2G1 and 7B9-9D11 + 2G1 cocktails that picked from the VSV-SARS-CoV-2 system efficiently neutralized all current variants of concern and variants of interest including the most recent variants Delta and Omicron, as well as SARS-CoV-1. Our results highlight the feasibility of using the VSV- SARS-CoV-2 system to develop SARS-CoV-2 antibody cocktails and provide a reference for the clinical selection of therapeutic strategies to address the mutational escape of SARS-CoV-2.
Keywords: SARS-CoV-2; antibody; vesicular stomatitis virus; variant; neutralization

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